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PAT-1251

Glpbio
Catalog No:GC30112-5mg CAS No.:2007885-39-2 MDLNo: Brand:Glpbio purity: 特性: Purpose:PAT-1251是一种有效的,选择性的,可口服的赖氨酰氧化酶样蛋白2(LOXL2)抑制剂,对hLOXL2和hLOXL3的IC50值分别为0.71和1.17μM,同时对小鼠、大鼠和狗LOXL2的抑制作用很强,IC50值分别为0.10,0.12和0.16μM;PAT-1251已经进入临床开发,有治疗多种纤维性疾病的潜力。DMSO : ≥ 130 mg/mL (325.54 mM)
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