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JNJ-10229570

Glpbio
Catalog No:GC30194-5mg CAS No.:524923-88-4 MDLNo: Brand:Glpbio purity: 特性: Purpose:JNJ-10229570是肾上腺皮质受体1(MC1R)和肾上腺皮质受体5(MC5R)的拮抗剂,可抑制皮脂腺分化和皮质特异性脂质的产生,其抑制125I-NDP-α-MSH和人类细胞中MC1R和MC5R结合的IC50值分别为270nM和200nM。DMSO : 62.5 mg/mL (160.47 mM; Need ultrasonic)
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