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YF-2

Glpbio
Catalog No:GC31099-10mg CAS No.:1311423-89-8 MDLNo: Brand:Glpbio purity: 特性: Purpose:YF-2是一种高度选择性、可透过血脑屏障的组蛋白乙酰转移酶(histoneacetyltransferase)激动剂,能够在海马区乙酰化H3,对CBP,PCAF和GCN5的EC50值分别为2.75μM,29.04μM和49.31μM,对HDAC无作用。具有抗肿瘤和抗阿尔滋海默症的活性。DMSO : ≥ 125 mg/mL (290.12 mM);H2O : < 0.1 mg/mL (insoluble)
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