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ACT-709478

Glpbio
Catalog No:GC31100-10mM(1mLinDMSO) CAS No.:1838651-58-3 MDLNo: Brand:Glpbio purity: 特性: Purpose:ACT-709478是一种有效、选择性、可口服、可透过血脑屏障的T型电压门控钙通道(T-typecalciumchannel)阻滞剂,对Cav3.1,Cav3.2,Cav3.3,Cav1.2的IC50值分别为6.4,18,7.5和2410nM。ACT-709478对大鼠、小鼠、狗和猕猴的T-typecalciumchannel都有作用,物种差异不大。ACT-709478可用于全身性癫痫的研究。DMSO : ≥ 125 mg/mL (293.83 mM)
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