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Abrocitinib (PF-04965842)

Glpbio
Catalog No:GC32023-10mM(1mLinDMSO) CAS No.:1622902-68-4 MDLNo: Brand:Glpbio purity: 特性: Purpose:Abrocitinib(PF-04965842)是一种有效、可口服、选择性的JAK1抑制剂,对JAK1和JAK2的IC50值分别为29和803nM。Abrocitinib(PF-04965842)可抑制TYK2的活性(IC50,1.253μM)和刺激后STAT1,STAT3和STAT5的磷酸化水平。可用于自身免疫症的研究。DMSO : 125 mg/mL (386.51 mM; Need ultrasonic)
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