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TAK-220

Glpbio
Catalog No:GC32135-10mM(1mLinDMSO) CAS No.:333994-00-6 MDLNo: Brand:Glpbio purity: 特性: Purpose:TAK-220是一种选择性的,可口服的CCR5拮抗剂,能够抑制RANTES,MIP-1α与CCR5结合,IC50值分别为3.5nM和1.4nM,但是对CCR1,CCR2b,CCR3,CCR4或者CCR7无作用;TAK-220也可选择性地抑制HIV-1,在外周单核细胞中,EC50值分别为1.2nM(HIV-1KK),0.72nM(HIV-1CTV),1.DMSO : ≥ 50 mg/mL (90.39 mM)
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