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SEL120-34A monohydrochloride

Glpbio
Catalog No:GC34355-10mM(1mLinDMSO) CAS No.: MDLNo: Brand:Glpbio purity: 特性: Purpose:SEL120-34Amonohydrochloride是一种选择性的,ATP-竞争性的CDK8抑制剂,对CDK8/CycC和CDK19/CycC复合物的IC50值分别为4.4nM和10.4nM,对CDK8的Kd值为3nM。SEL120-34Amonohydrochloride对CDK9的作用很弱,计算的IC50值为1070nM,DMSO : 13 mg/mL (28.85 mM; Need ultrasonic)
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