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(R)-BAY1238097

Glpbio
Catalog No:GC34443-50mg CAS No.:1564269-85-7 MDLNo: Brand:Glpbio purity: 特性: Purpose:(R)-BAY1238097是BAY1238097的低活性R型异构体。BAY1238097是一种有效的、BET与组蛋白结合的选择性抑制剂,通过下调c-Myc水平及下游转录组,在AML(急性髓性白血病)和MM(多发性骨髓瘤)模型中表现出较强的抗增殖活性。DMSO : 150 mg/mL (332.18 mM; Need ultrasonic);H2O : < 0.1 mg/mL (insoluble)
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