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GGTI-2418

Glpbio
Catalog No:GC34592-5mg CAS No.:501010-06-6 MDLNo: Brand:Glpbio purity: 特性: Purpose:GGTI-2418是一种高效,竞争性和选择性的香叶基香叶基转移酶I(GGTaseI)抑制剂。GGTI-2418抑制GGTaseI和FTase活性,IC50分别为9.5nM和53μM。GGTI-2418还增强p27(Kip1)并诱导乳腺肿瘤显着消退。DMSO : 125 mg/mL (283.11 mM; Need ultrasonic)
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