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SGC-iMLLT

Glpbio
Catalog No:GC34778-50mg CAS No.:2255338-25-9 MDLNo: Brand:Glpbio purity: 特性: Purpose:SGC-iMLLT是一种有效、选择性的MLLT1/3-histone相互作用抑制剂,与MLLT1YD上的Kac/Kcr结合位点结合,对MLLT1YD(ENL/YEATS1)(IC50,0.26 μM;Kd,0.129 μM)和MLLT3YD(AF9/YEATS3)(Kd,0.077 μM)具有很高的亲和性。DMSO : 83.33 mg/mL (214.51 mM; Need ultrasonic);H2O : < 0.1 mg/mL (insoluble)
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