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CAY10471 Racemate

Glpbio
Catalog No:GC35620-10mg CAS No.:844639-57-2 MDLNo: Brand:Glpbio purity: 特性: Purpose:CAY10471 Racemate (TM30089 Racemate) 是一种有效、高度选择性的前列腺素 D2 受体 (CRTH2) 拮抗剂,对 hCRTH2 的 Ki 值为 0.6 nM,对其选择性远高于人血栓素 A2 受体 TP (Ki,10000 nM) 或 PGD2 受体 DP (Ki,1200 nM)。CAY10471 Racemate 对小鼠和大鼠的同源 CRTH2 也具有拮抗作用。DMSO: 150 mg/mL (360.17 mM)
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