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CX-5461 dihydrochloride

Glpbio
Catalog No:GC35761-5mg CAS No.: MDLNo: Brand:Glpbio purity: 特性: Purpose:CX-5461 dihydrochloride 是一种有效的,可口服的 Pol I 介导的 rRNA synthesis 抑制剂,在 HCT-116,A375 和 MIA PaCa-2 细胞中,IC50 值分别为 142 nM,113 nM 和 54 nM,对 Pol II 作用不大 (IC50 ≥25 μM)。H2O: ≥ 25 mg/mL (42.62 mM)
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