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DDD107498 succinate

Glpbio
Catalog No:GC35820-10mg CAS No.: MDLNo: Brand:Glpbio purity: 特性: Purpose:DDD107498 succinate (DDD-498 succinate) 是一种有效、可口服的抗疟疾 (antimalarial) 剂,能够抑制寄生虫生命周期的多个阶段,对 P. falciparum 3D7 的 EC50 值为 1 nM。DDD107498 succinate (DDD-498 succinate) 通过靶作用于 eEF2/CaMKIII 来抑制蛋白合成,对 WT-PfeEF2 的 EC50 值为 2 nM。DMSO: 135 mg/mL (232.50 mM)
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