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ERK5-IN-2

Glpbio
Catalog No:GC36002-25mg CAS No.:1888305-96-1 MDLNo: Brand:Glpbio purity: 特性: Purpose:ERK5-IN-2 是一种具有口服活性,亚微摩尔效力,选择性的 ERK5 抑制剂,对 ERK5 和 ERK5 MEF2D 的 IC50s 分别是 0.82 μM,3 μM。ERK5-IN-2 不与 BRD4 溴结构域相互作用。ERK5-IN-2 抑制肿瘤异种移植生长和 碱性成纤维细胞生长因子 (bFGF) 驱动的基质胶塞血管的生成。DMSO: 250 mg/mL (644.01 mM)
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