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FGTI-2734

Glpbio
Catalog No:GC36038-5mg CAS No.:1247018-19-4 MDLNo: Brand:Glpbio purity: 特性: Purpose:FGTI-2734 是 RAS C-末端法尼基转移酶 (FT) 和香叶烯基转移酶-1 (GGT) 抑制剂,对 FT 和 GGT 的 IC50s 分别为 250 nM和 520 nM。 FGTI-2734 可以阻断 KRAS 的膜定位,从而解决 KRAS 耐药性问题,并抑制突变的 KRAS 胰腺肿瘤。DMSO: 50 mg/mL (97.92 mM)
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