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LOC14

Glpbio
Catalog No:GC36473-5mg CAS No.:877963-94-5 MDLNo: Brand:Glpbio purity: 特性: Purpose:LOC14 是蛋白质二硫键异构酶 (PDI) 抑制剂 (EC50=500 nM; Kd=62 nM)。LOC14 在小鼠肝微粒体和血浆中表现出高稳定性,低内在微粒体清除率和低血浆蛋白结合。LOC14 抑制 PDIA3 活性,降低肺上皮细胞中 HA 的分子内二硫键和随后的寡聚化。DMSO: 25 mg/mL (78.76 mM)
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