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PT2977

Glpbio
Catalog No:GC37034-1mg CAS No.:1672668-24-4 MDLNo: Brand:Glpbio purity: 特性: Purpose:PT2977 是一种口服有效的,选择性 HIF-2α 抑制剂,IC50 为 9 nM。PT2977 作为第二代 HIF-2α 抑制剂,可提高效力并改善药代动力学特征。PT2977 是一种潜在的治疗透明细胞肾细胞癌 (ccRCC) 和 VHL 疾病的方法。DMSO: 50 mg/mL (130.43 mM)
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