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RU.521

Glpbio
Catalog No:GC37570-100mg CAS No.:2262452-06-0 MDLNo: Brand:Glpbio purity: 特性: Purpose:RU.521 (RU320521) 是一种有效的 dsDNA 和 cGAS 抑制剂,对 dsDNA 的 IC50 为700 nM。 RU.521 抑制 cGAS 介导的干扰素上调,抑制 dsDNA 依赖性激活。 RU.521 在环状 GMP-AMP 合酶介导的信号传导的细胞测定中具有活性和选择性,并且降低来自 Aicardi-Goutières 综合征小鼠模型的巨噬细胞中干扰素的组成型表达。DMSO: ≥ 125 mg/mL (301.04 mM)
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