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Taccalonolide A

Glpbio
Catalog No:GC37715-5mg CAS No.:108885-68-3 MDLNo: Brand:Glpbio purity: 特性: Purpose:Taccalonolide A 是一种微管稳定剂,是从 Tacca chantrieri 中分离得到的类固醇,具有细胞毒性和抗疟活性。Taccalonolide A 能引起 G2-M 期滞留、Bcl-2 磷酸化,并引发细胞凋亡。Taccalonolide A 在体外对过表达 p 糖蛋白 (Pgp)、多药耐药蛋白 7 (MRP7) 的细胞系具有显著的抑制作用,抑制SK-OV-3细胞生长的 IC50 值为 622 nM。Soluble in DMSO
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