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TAK-960 dihydrochloride

Glpbio
Catalog No:GC37725-50mg CAS No.: MDLNo: Brand:Glpbio purity: 特性: Purpose:TAK-960 dihydrochloride 是一种有效的,可口服的,选择性的 polo-like kinase 1 (PLK1) 抑制剂,在 10 μM ATP 的条件下,IC50 值为 0.8 nM;TAK-960 dihydrochloride 同时对 PLK2 和 PLK3 也有抑制作用,IC50 值分别为 16.9 和 50.2 nM。DMSO: ≥ 98.57 mg/mL (155.35 mM)
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