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TAK-960 hydrochloride

Glpbio
Catalog No:GC37726-100mg CAS No.:1137868-96-2 MDLNo: Brand:Glpbio purity: 特性: Purpose:TAK-960 hydrochloride 是一种有效的,可口服的,选择性的 polo-like kinase 1 (PLK1) 抑制剂,在 10 μM ATP 的条件下,IC50 值为 0.8 nM;TAK-960 hydrochloride 同时对 PLK2 和 PLK3 也有抑制作用,IC50 值分别为 16.9 和 50.2 nM。。Soluble in DMSO
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