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NS13001

Glpbio
Catalog No:GC38200-10mg CAS No.:1063331-94-1 MDLNo: Brand:Glpbio purity: 特性: Purpose:NS13001 是一种有效的、选择性的、具有口服活性 SK channels (小电导钙激活钾通道) 正向变构调节剂。NS13001 对 SK2 和 SK3 通道的 EC50 分别为 1.8 μM 和 0.14 μM。NS13001 有望作为治疗脊髓小脑共济失调 2 型 (SCA2) 和可能的其他小脑共济失调的潜在治疗剂。DMSO: 100 mg/mL (282.64 mM); H2O: < 0.1 mg/mL (insoluble)
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