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BMS-986020 sodium

Glpbio
Catalog No:GC38470-100mg CAS No.:1380650-53-2 MDLNo: Brand:Glpbio purity: 特性: Purpose:BMS-986020 sodium 是高亲和力溶血磷脂酸受体 1 (LPA1) 拮抗剂。BMS-986020 sodium 抑制胆汁酸和磷脂转运蛋白,抑制 BSEP,MRP4 和 MDR3,IC50 值分别为 4.8 μM,6.2 μM 和 7.5 μM。BMS-986020 sodium 用于治疗特发性肺纤维化 (IPF)。DMSO: 150 mg/mL (297.32 mM); H2O: < 0.1 mg/mL (insoluble)
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