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Ilorasertib hydrochloride

Glpbio
Catalog No:GC38519-10mg CAS No.:1847485-91-9 MDLNo: Brand:Glpbio purity: 特性: Purpose:Ilorasertib hydrochloride (ABT-348 hydrochloride) 是一种有效、ATP 竞争性的多靶点激酶抑制剂,可抑制 Aurora C,Aurora B 和 Aurora A 的活性,IC50 值分别为 1 nM,7 nM 和 120 nM。Ilorasertib hydrochloride (ABT-348 hydrochloride) 同时抑制 RET,PDGFRβ 和 Flt1 的活性,IC50 值分别为 7 nM,3 nM 和 32 nM。DMSO: 41.67 mg/mL (79.37 mM)
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