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PXS-5153A monohydrochloride

Glpbio
Catalog No:GC38583-5mg CAS No.: MDLNo: Brand:Glpbio purity: 特性: Purpose:PXS-5153A monohydrochloride 是一种有效的、选择性的、具有口服活性和快速起效的赖氨酰氧化酶 2/3 (LOXL2/LOXL3) 的双抑制剂,对几乎所有哺乳动物LOXL2的IC50 均< 40 nM,对人类LOXL3 的IC50 为63 nM。PXS-5153A monohydrochloride 可减少交联,改善纤维化。DMSO: 250 mg/mL (569.54 mM)
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