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PTC596

Glpbio
Catalog No:GC38592-10mg CAS No.:1610964-64-1 MDLNo: Brand:Glpbio purity: 特性: Purpose:PTC596 是一种口服活性和选择性的 B 细胞特异性莫洛尼氏鼠白血病病毒整合位点 1 (BMI-1) 抑制剂。PTC596 靶向肿瘤细胞和癌症干细胞 (CSC) 均表达的 BMI1,并诱导 BMI1 过度磷酸化,从而导致其降解。PTC596 可下调 MCL-1 并诱导急性髓系白血病祖细胞中不依赖 p53 的线粒体凋亡。DMF: 30 mg/ml,DMSO: 30 mg/ml,Ethanol: 5 mg/ml
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