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Lanraplenib succinate

Glpbio
Catalog No:GC38630-1mg CAS No.:1800047-00-0 MDLNo: Brand:Glpbio purity: 特性: Purpose:Lanraplenib succinate (GS-9876 succinate) 是一种高度选择性的口服 SYK 抑制剂 (IC50=9.5 nM) ,用于治疗炎症性疾病。Lanraplenib succinate (GS-9876 succinate) 通过糖蛋白 VI (GPVI) 受体抑制血小板中的 SYK 活性,而不会延长猴子或人类的出血时间 (BT)。DMSO: 83.33 mg/mL (134.26 mM)
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