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KDOAM-25 citrate

Glpbio
Catalog No:GC38709-100mg CAS No.: MDLNo: Brand:Glpbio purity: 特性: Purpose:KDOAM-25 citrate 是有效,高选择性的 KDM5 抑制剂,对 KDM5A,KDM5B,KDM5C,KDM5D 的 IC50 分别为 71 nM,19 nM,69 nM,69 nM。KDOAM-25 citrate 可增加转录起始位点的整体 H3K4 甲基化,并损害多发性骨髓瘤 MM1S 细胞的增殖。DMSO: 200 mg/mL (400.39 mM)
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