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AS2863619

Glpbio
Catalog No:GC38736-10mg CAS No.:2241300-51-4 MDLNo: Brand:Glpbio purity: 特性: Purpose:AS2863619 可以将抗原特异性效应子/记忆 T 细胞转换为 Foxp3+ 调节性 T (Treg) 细胞,以治疗各种免疫疾病。AS2863619 是一种有效的口服的细胞周期蛋白依赖性激酶 8 (CDK8) 和 CDK19 抑制剂,IC50 分别为 0.61 nM 和 4.28 nM。AS2863619 抑制 CDK8/19 可增强 STAT5 的激活,从而激活 Foxp3 基因。DMSO: 250 mg/mL (616.92 mM)
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