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CKI-7

Glpbio
Catalog No:GC38755-1mg CAS No.:120615-25-0 MDLNo: Brand:Glpbio purity: 特性: Purpose:CKI-7 是一种有效且 ATP 竞争性的酪蛋白激酶 1 (CK1) 抑制剂,IC50 为 6 μM,Ki 为 8.5 μM。CKI-7 选择性抑制 Cdc7 激酶,还抑制 SGK,S6K1 以及 MSK1。CKI-7 对酪蛋白激酶 II 和其他蛋白激酶的作用弱得多。DMSO: 25 mg/mL (87.49 mM)
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