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GSK-25

Glpbio
Catalog No:GC38791-1mg CAS No.:874119-56-9 MDLNo: Brand:Glpbio purity: 特性: Purpose:GSK-25 是一种有效的、选择性的,具有口服活性的 ROCK1 抑制剂 (IC50=7 nM)。GSK-25 对 31 种激酶以及 RSK1 和 p70S6K 保持良好的选择性 (RSK1: IC50=398 nM, p70S6K: IC50=1 μM)。GSK-25 可抑制 P450 (CYP2C9、CYP2D6、CYP3A4的IC50 分别为2.5、5.2、2.5 μM)。DMSO: 100 mg/mL (194.81 mM)
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