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Lapaquistat acetate

Glpbio
Catalog No:GC38807-5mg CAS No.:189060-13-7 MDLNo: Brand:Glpbio purity: 特性: Purpose:Lapaquistat acetate (TAK-475) 是一种角鲨烯合酶 (squalene synthase) 抑制剂,可阻止法呢基二磷酸酯 (FPP) 转化为角鲨烯。Lapaquistat acetate (TAK-475) 最初旨在用于甲羟戊酸激酶缺乏症 (MKD),可有效降低低密度脂蛋白胆固醇,但可能引起肝脏损害。DMSO: 46 mg/mL (71.30 mM)
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