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TRAF-STOP inhibitor 6877002

Glpbio
Catalog No:GC38868-10mg CAS No.:433249-94-6 MDLNo: Brand:Glpbio purity: 特性: Purpose:TRAF-STOP inhibitor 6877002,一种抑制 CD40-TRAF6 相互作用的选择性抑制剂,从专利 WO2014033122A1 中获得,抑制 RAW 细胞中 NF-κB 活化,化合物VII。TRAF-STOP 6877002 可阻止小鼠中已发生的动脉粥样硬化恶化,减少白细胞募集并减少巨噬细胞活化;减少动脉粥样硬化斑块中的巨噬细胞增殖。DMSO: 125 mg/mL (497.37 mM)
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