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LCH-7749944

Glpbio
Catalog No:GC39209-10mg CAS No.:796888-12-5 MDLNo: Brand:Glpbio purity: 特性: Purpose:LCH-7749944 (GNF-PF-2356) 是一种有效的 PAK4 抑制剂,IC50 为 14.93 μM。LCH-7749944通过下调 PAK4/c-Src/EGFR/cyclin D1 途径有效抑制人胃癌细胞的增殖,并诱导凋亡 (apoptosis)。DMSO: 250 mg/mL (713.45 mM)
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