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GSK2798745

Glpbio
Catalog No:GC39387-10mg CAS No.:1419609-94-1 MDLNo: Brand:Glpbio purity: 特性: Purpose:GSK2798745 是一流的,高效的,选择性的且具有口服活性的 瞬时受体电位香草酸 4 (TRPV4) 离子通道阻断剂,对于 hTRPV4 和 rTRPV4 的 IC50 值分别为 1.8 和 1.6 nM。GSK2798745 用于治疗与充血性心力衰竭相关的肺水肿的研究。DMSO: 250 mg/mL (542.85 mM)
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