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PDK4-IN-1 hydrochloride

Glpbio
Catalog No:GC39500-100mg CAS No.:2310262-11-2 MDLNo: Brand:Glpbio purity: 特性: Purpose:PDK4-IN-1 hydrochloride 是一种蒽醌衍生物,也是一种有效的,口服活性的丙酮酸脱氢酶激酶 4 (PDK4) 抑制剂,IC50 值为 84 nM。PDK4-IN-1 hydrochloride 有效抑制细胞转化和细胞增殖并诱导细胞凋亡 (apoptosis)。PDK4-IN-1 hydrochloride 具有抗糖尿病,抗癌和抗过敏作用。DMSO: 125 mg/mL (317.36 mM)
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