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PF-04634817 succinate

Glpbio
Catalog No:GC39501-1mg CAS No.:2140301-98-8 MDLNo: Brand:Glpbio purity: 特性: Purpose:PF-0463481 succinate 是一种有效的具有口服活性的双效 CCR2/CCR5 拮抗剂,对人和啮齿类动物的 CCR2 效价相当 (rat IC50=20.8 nM),对 CCR2 的效价是 CCR5 的 10-20 倍 (rat IC50=470 nM)。PF-0463481 succinate 安全、耐受性好,有潜力用于研究糖尿病肾病。Soluble in DMSO
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