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TED-347

Glpbio
Catalog No:GC39540-1mg CAS No.:2378626-29-8 MDLNo: Brand:Glpbio purity: 特性: Purpose:TED-347 是一种有效,不可逆且共价的 YAP-TEAD 蛋白质-蛋白质相互作用变构抑制剂,对 TEAD4&;Yap1 蛋白质-蛋白质相互作用的 EC50 为 5.9 μM。TED-347 与 TEAD4 中央口袋内的 Cys-367 特异性共价结合,Ki 为 10.3 μM。TED-347 可以阻断 TEAD 的转录活性,并且具有抗肿瘤活性。DMSO: 250 mg/mL (796.94 mM)
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