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BPN-15606

Glpbio
Catalog No:GC39566-50mg CAS No.:1914989-49-3 MDLNo: Brand:Glpbio purity: 特性: Purpose:BPN-15606 是一种高效的口服活性 γ-secretase 调节剂 (GSM),可减弱 SHSY5Y 神经母细胞瘤细胞产生 Aβ42 和 Aβ40 的作用,IC50 值分别为 7 nM 和 17 nM。BPN-15606 显着降低大鼠和小鼠中枢神经系统中的 Aβ42 和 Aβ40 水平。BPN-15606 具有良好的 PK/PD 特性,包括生物利用度,半衰期和清除率。DMSO: 100 mg/mL (238.97 mM)
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