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BRD5529

Glpbio
Catalog No:GC39622-5mg CAS No.:1358488-78-4 MDLNo: Brand:Glpbio purity: 特性: Purpose:BRD5529 是一种选择性 CARD9-E3 泛素连接酶 TRIM62 蛋白-蛋白相互作用抑制剂,IC50 为 8.6 μM。BRD5529 选择性地直接与 CARD9 结合,破坏 TRIM62 募集,抑制 TRIM62 介导的 CARD9 泛素化和激活,并在依赖 CARD9 的途径中表现出细胞活性和选择性。DMSO: 250 mg/mL (537.01 mM)
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