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BI-9321 trihydrochloride

Glpbio
Catalog No:GC39663-10mg CAS No.:2387510-87-2 MDLNo: Brand:Glpbio purity: 特性: Purpose:BI-9321 trihydrochloride 是一种有效的,选择性的,具有细胞活性的 NSD3-PWWP1 拮抗剂,Kd 值为 166 nM。BI-9321 对 NSD2-PWWP1 和 NSD3-PWWP2 无效。BI-9321 trihydrochloride 在 U2OS 细胞中特异性破坏 NSD3-PWWP1 与组蛋白相互作用,IC50 为 1.2 μM。DMSO: 250 mg/mL (532.13 mM)
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