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VU0134992 hydrochloride

Glpbio
Catalog No:GC39667-50mg CAS No.:1052515-91-9 MDLNo: Brand:Glpbio purity: 特性: Purpose:VU0134992 hydrochloride 是第一个亚型偏好的,具有口服活性和选择性的内向整流钾通道 Kir4.1 阻滞剂,IC50 值为 0.97 μM。VU0134992 hydrochloride 在 -120 mV 时,对同分 Kir4.1 比 Kir4.1/5.1 共分通道 (IC50=9 μM) 高出 9 倍的选择性。DMSO: 250 mg/mL (558.24 mM)
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Chemical safety data sheet(MSDS)

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