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3-Hydroxy Midostaurin

Glpbio
Catalog No:GC39689-100mg CAS No.:179237-49-1 MDLNo: Brand:Glpbio purity: 特性: Purpose:3-Hydroxy Midostaurin (CGP 52421) 是 PKC412 的代谢产物,可有效抑制 FMS 样酪氨酸激酶 3 (FLT3) 自磷酸化,在培养基和血浆中的 IC50 分别为 132 nM 和 9.8 μM。与 PKC412 相比,3-Hydroxy Midostaurin 的选择性较低,但细胞毒性更高。Soluble in DMSO
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