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Facinicline hydrochloride

Glpbio
Catalog No:GC39748-100mg CAS No.:677305-02-1 MDLNo: Brand:Glpbio purity: 特性: Purpose:Facinicline hydrochloride (RG3487 hydrochloride) 是具有口服活性的烟碱 α7 receptor 部分激动剂,对人nAChR 的 Ki 值为 6 nM。Facinicline hydrochloride (RG3487 hydrochloride) 可改善啮齿类动物的认知和感觉运动门控。Facinicline hydrochloride (RG3487 hydrochloride) 对5-HT3 受体 (拮抗剂)的Ki 值为 1.2 nM。DMSO: 125 mg/mL (407.44 mM); Methanol: 25 mg/mL (81.49 mM)
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