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Brexpiprazole S-oxide

Glpbio
Catalog No:GC60662-5mg CAS No.:1191900-51-2 MDLNo:C25H27N3O3S Brand:Glpbio purity: 特性: Purpose:BrexpiprazoleS-oxide(DM-3411)是Brexpiprazole的主要代谢产物,并通过细胞色素P4503A4(CYP3A4)代谢。Brexpiprazole是一种非典型抗精神病药,是人5-HT1A和多巴胺受体的部分激动剂,Ki分别为0.12nM和0.3nM。Brexpiprazole也是5-HT2A受体的拮抗剂,Ki为0.47nM。
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Product Overview
Product Name Brexpiprazole S-oxide
CAS1191900-51-2
MW449.57
MDLC25H27N3O3S
Storage conditionPowder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
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