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Imatinib Impurity E

Glpbio
Catalog No:GC60931-1mg CAS No.:1365802-18-1 MDLNo:C52H48N12O2 Brand:Glpbio purity: 特性: Purpose:ImatinibImpurityE是Imatinib的杂质。Imatinib是一种口服生物可用的酪氨酸激酶抑制剂,可选择性抑制BCR/ABL,v-Abl,PDGFR,c-kit激酶活性。Imatinib(STI571)靠近ATP结合位点结合,将其锁定在封闭或自我抑制的构象中,因此半竞争性抑制蛋白质的酶活性。Imatinib还抑制SARS-CoV和MERS-CoV。
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